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3ZON

Human TYK2 pseudokinase domain bound to a kinase inhibitor

Summary for 3ZON
Entry DOI10.2210/pdb3zon/pdb
DescriptorNON-RECEPTOR TYROSINE-PROTEIN KINASE TYK2, 5-PHENYL-2-UREIDOTHIOPHENE-3-CARBOXAMIDE (3 entities in total)
Functional Keywordstransferase, jak
Biological sourceHOMO SAPIENS (HUMAN)
Total number of polymer chains1
Total formula weight37667.81
Authors
Elkins, J.M.,Wang, J.,Krojer, T.,Savitsky, P.,Chalk, R.,Daga, N.,Salah, E.,Berridge, G.,Picaud, S.,von Delft, F.,Bountra, C.,Edwards, A.,Knapp, S. (deposition date: 2013-02-22, release date: 2013-04-10, Last modification date: 2023-12-20)
Primary citationElkins, J.M.,Wang, J.,Krojer, T.,Savitsky, P.,Chalk, R.,Daga, N.,Salah, E.,Berridge, G.,Picaud, S.,von Delft, F.,Bountra, C.,Edwards, A.,Knapp, S.
Human Tyk2 Pseudokinase Domain Bound to a Kinase Inhibitor
To be Published,
Experimental method
X-RAY DIFFRACTION (2.15 Å)
Structure validation

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